Exposing Novel Kinase Polypharmacology and Drug Escape Mechanisms in Cells With NanoBRET

Time: 11:45 am
day: Day One


  • Enabling live cell kinase profiling: Exploring the landscape of DDR kinase inhibitors in cells
  • Kinome-wide live cell profiling reveals novel interactions for type II kinase inhibitors
  • Protomer selectivity of RAF dimer inhibitors informs on the mechanism of inhibition within the RAS-RAF signalosome