Monitoring Continuous Enzyme Activity with Fluorogenic Sensor Assays Enables Data-Rich Decisions for Improved Kinase & Phosphatase Drug Discovery
Time: 2:15 pm
day: Day One
Details:
- Advantages of PhosphoSens® technology as a continuous activity assay (a progress curve in every well)
- Kinome selectivity profiling at low or high ATP with insight into compound dependent kinetics and MOA
- Deep characterization of kinase inhibitor potency for reversible or irreversible inhibitors