Monitoring Continuous Enzyme Activity with Fluorogenic Sensor Assays Enables Data-Rich Decisions for Improved Kinase & Phosphatase Drug Discovery

Time: 2:15 pm
day: Day One

Details:

  • Advantages of PhosphoSens® technology as a continuous activity assay (a progress curve in every well)
  • Kinome selectivity profiling at low or high ATP with insight into compound dependent kinetics and MOA
  • Deep characterization of kinase inhibitor potency for reversible or irreversible inhibitors

Speakers: